AhR Agonists
| Cat.No. | Product Name | Information | Product Use Citations | Product Validations |
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| S7711 | CH-223191 | CH-223191 is a potent and specific aryl hydrocarbon receptor (AhR) antagonist with IC50 of 30 nM. |
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| S2858 | Stemregenin 1 (SR1) | StemRegenin 1 (SR1) is an aryl hydrocarbon receptor (AhR) inhibitor with IC50 of 127 nM in a cell-free assay. |
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| S8995 | BAY 2416964 | BAY 2416964 (compound 192) is a potent and orally active antagonist of aryl hydrocarbon receptor (AhR) with an IC50 of 341 nM. This compound has the potential in the treatment of solid tumours. |
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| S6560 | PDM2 | PDM2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist. |
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| S6926 | GNF351 | GNF351 is a potent antagonist of the aryl hydrocarbon receptor (AHR). This compound interacts directly with the AHR ligand binding pocket and competes with a well-characterised photoaffinity AHR ligand for binding to the AHR with an IC50 of 62 nM. |
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| S0155 | PDM-11 | PDM-11 is a derivative of resveratrol that exhibits stronger antagonist affinity for arylhydrocarbon receptors (AhR) than resveratrol, without any affinity for the estrogen receptor. | ||
| S1177 | PD 98059 | PD98059 is a non-ATP competitive MEK inhibitor with IC50 of 2 μM in a cell-free assay, specifically inhibits MEK-1-mediated activation of MAPK; does not directly inhibit ERK1 or ERK2. PD98059 is a ligand for the aryl hydrocarbon receptor (AHR) and functions as an AHR antagonist. |
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